FALESIEDI, MARTA
FALESIEDI, MARTA
100019 - Dipartimento di chimica e chimica industriale
A family of nitrogen-containing heterocycles as sirtuin inhibitors: synthesis and invitro biological evaluation
2024-01-01 Falesiedi, M.; Scarano, N.; Grossi, G.; Carbone, A.; Brullo, C.; Musumeci, Francesca; Bruzzone, S.; Cichero, E.; Schenone, S.
Approaching Gallium-68 radiopharmaceuticals for tumor diagnosis: a Medicinal Chemist’s perspective
2025-01-01 Musumeci, Francesca; Fasce, Alessandro; Falesiedi, Marta; Oleari, Federica; Grossi, Giancarlo; Carbone, Anna; Schenone, Silvia
Combining repositioning and de novo synthesis of pyrazolo[3,4-d]pyrimidines to discover potent SIRT-2 inhibitors
2024-01-01 Falesiedi, Marta; Scarano, Naomi; Grossi, Giancarlo; Carbone, Anna; Brullo, Chiara; Musumeci, Francesca; Bruzzone, Santina; Cichero, Elena; Schenone, Silvia.
DESIGN AND SYNTHESIS OF TRIAZINE DERIVATIVES AS POTENTIAL SIRT2 INHIBITORS: A MOLECULAR SIMPLIFICATION APPROACH
2025-01-01 Oleari, F.; Musumeci, F.; Falesiedi, M.; Nicolini, F.; Salis, A.; Cichero, E.; Bruzzone, S.; Schenone, S.
From pyrazolo[3,4-d]pyrimidine to triazine scaffold: synthesis of a new family of SIRT-2 inhibitors
2025-01-01 Oleari, F.; Musumeci, F.; Falesiedi, M.; Nicolini, F.; Salis, A.; Cichero, E.; Bruzzone, S.; Schenone, S.
Halloysite Nanotube-Based Delivery of Pyrazolo[3,4-d]pyrimidine Derivatives for Prostate and Bladder Cancer Treatment
2024-01-01 Massaro, Marina; Ciani, Rebecca; Grossi, Giancarlo; Cavallaro, Gianfranco; de Melo Barbosa, Raquel; Falesiedi, Marta; Fortuna, Cosimo G.; Carbone, Anna; Schenone, Silvia; Sánchez-Espejo, Rita; Viseras, César; Vago, Riccardo; Riela, Serena
PYRAZOLO[3,4-d]PYRIMIDINE DERIVATIVES AS SIRTUIN INHIBITORS: DESIGN, SYNTHESIS AND PRELIMINARY in vitro EVALUATION
2024-01-01 Falesiedi, Marta; Grossi, Giancarlo; Carbone, Anna; Brullo, Chiara; Musumeci, Francesca; Bruzzone, Santina; Cichero, Elena; Schenone, Silvia
Pyrazolo[3,4-d]pyrimidines as Sirtuin Inhibitors: A Preliminary Synthetic and Biological Study
2025-01-01 Falesiedi, Marta; Scarano, Naomi; Grossi, Giancarlo; Carbone, Anna; Brullo, Chiara; Musumeci, Francesca; Bruzzone, Santina; Cichero, Elena; Schenone, Silvia
Small Molecule Tyrosine Kinase Inhibitors (TKIs) for Glioblastoma Treatment
2024-01-01 Frumento, Davide; Grossi, Giancarlo; Falesiedi, Marta; Musumeci, Francesca; Carbone, Anna; Schenone, Silvia
SYNTHESIS AND BIOLOGICAL EVALUATION OF NEW 4-AMINO-PYRAZOLO[3,4-d]PYRIMIDINES AS POTENTIAL SRC KINASE INHIBITORS
2023-01-01 Falesiedi, M.; Cianciusi, A.; Carbone, A.; Musumeci, F.; Schenone, S.; Angelucci, A.; Sabetta, S.; Maga, G.; Crespan, E.
Targeting Sirtuins with Pyrazolo[3,4-d]pyrimidines: A Synthetic and Biological Feasibility Study
2025-01-01 Falesiedi, M.; Scarano, N.; Grossi, G.; Carbone, A.; Musumeci, F.; Bruzzone, Santina; Cichero, E.; Schenone, S.
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| A family of nitrogen-containing heterocycles as sirtuin inhibitors: synthesis and invitro biological evaluation | 1-gen-2024 | Falesiedi, M.; Scarano, N.; Grossi, G.; Carbone, A.; Brullo, C.; Musumeci, Francesca; Bruzzone, S.; Cichero, E.; Schenone, S. | |
| Approaching Gallium-68 radiopharmaceuticals for tumor diagnosis: a Medicinal Chemist’s perspective | 1-gen-2025 | Musumeci, Francesca; Fasce, Alessandro; Falesiedi, Marta; Oleari, Federica; Grossi, Giancarlo; Carbone, Anna; Schenone, Silvia | |
| Combining repositioning and de novo synthesis of pyrazolo[3,4-d]pyrimidines to discover potent SIRT-2 inhibitors | 1-gen-2024 | Falesiedi, Marta; Scarano, Naomi; Grossi, Giancarlo; Carbone, Anna; Brullo, Chiara; Musumeci, Francesca; Bruzzone, Santina; Cichero, Elena; Schenone, Silvia. | |
| DESIGN AND SYNTHESIS OF TRIAZINE DERIVATIVES AS POTENTIAL SIRT2 INHIBITORS: A MOLECULAR SIMPLIFICATION APPROACH | 1-gen-2025 | Oleari, F.; Musumeci, F.; Falesiedi, M.; Nicolini, F.; Salis, A.; Cichero, E.; Bruzzone, S.; Schenone, S. | |
| From pyrazolo[3,4-d]pyrimidine to triazine scaffold: synthesis of a new family of SIRT-2 inhibitors | 1-gen-2025 | Oleari, F.; Musumeci, F.; Falesiedi, M.; Nicolini, F.; Salis, A.; Cichero, E.; Bruzzone, S.; Schenone, S. | |
| Halloysite Nanotube-Based Delivery of Pyrazolo[3,4-d]pyrimidine Derivatives for Prostate and Bladder Cancer Treatment | 1-gen-2024 | Massaro, Marina; Ciani, Rebecca; Grossi, Giancarlo; Cavallaro, Gianfranco; de Melo Barbosa, Raquel; Falesiedi, Marta; Fortuna, Cosimo G.; Carbone, Anna; Schenone, Silvia; Sánchez-Espejo, Rita; Viseras, César; Vago, Riccardo; Riela, Serena | |
| PYRAZOLO[3,4-d]PYRIMIDINE DERIVATIVES AS SIRTUIN INHIBITORS: DESIGN, SYNTHESIS AND PRELIMINARY in vitro EVALUATION | 1-gen-2024 | Falesiedi, Marta; Grossi, Giancarlo; Carbone, Anna; Brullo, Chiara; Musumeci, Francesca; Bruzzone, Santina; Cichero, Elena; Schenone, Silvia | |
| Pyrazolo[3,4-d]pyrimidines as Sirtuin Inhibitors: A Preliminary Synthetic and Biological Study | 1-gen-2025 | Falesiedi, Marta; Scarano, Naomi; Grossi, Giancarlo; Carbone, Anna; Brullo, Chiara; Musumeci, Francesca; Bruzzone, Santina; Cichero, Elena; Schenone, Silvia | |
| Small Molecule Tyrosine Kinase Inhibitors (TKIs) for Glioblastoma Treatment | 1-gen-2024 | Frumento, Davide; Grossi, Giancarlo; Falesiedi, Marta; Musumeci, Francesca; Carbone, Anna; Schenone, Silvia | |
| SYNTHESIS AND BIOLOGICAL EVALUATION OF NEW 4-AMINO-PYRAZOLO[3,4-d]PYRIMIDINES AS POTENTIAL SRC KINASE INHIBITORS | 1-gen-2023 | Falesiedi, M.; Cianciusi, A.; Carbone, A.; Musumeci, F.; Schenone, S.; Angelucci, A.; Sabetta, S.; Maga, G.; Crespan, E. | |
| Targeting Sirtuins with Pyrazolo[3,4-d]pyrimidines: A Synthetic and Biological Feasibility Study | 1-gen-2025 | Falesiedi, M.; Scarano, N.; Grossi, G.; Carbone, A.; Musumeci, F.; Bruzzone, Santina; Cichero, E.; Schenone, S. |