IRIS
GROSSI, GIANCARLO
 Distribuzione geografica
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Continente #
EU - Europa 6.542
AS - Asia 21
SA - Sud America 4
NA - Nord America 1
Totale 6.568
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Nazione #
IT - Italia 6.542
CN - Cina 12
SG - Singapore 6
BR - Brasile 3
VN - Vietnam 3
AR - Argentina 1
US - Stati Uniti d'America 1
Totale 6.568
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Città #
Genova 3.657
Genoa 1.935
Rapallo 507
Vado Ligure 430
Bordighera 13
Beijing 4
Singapore 2
Ashburn 1
Bom Jesus da Lapa 1
Ho Chi Minh City 1
Huế 1
Phú Thọ 1
Santa Maria 1
Taquarana 1
Totale 6.555
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Nome #
1,2-Fused Pyrimidines. V. Synthesis of 1-Alkyl or Phenyl-2H-dipyrido-[1,2-a:2’, 3’-d]pyrimidine-2,5(1H)-diones 333
1,5-Benzodiazepines IX. A new route to substituted 4H-[1,2,4]triazolo[4,3-a][1,5]benzodiazepin-5-amines with analgesic and/or anti-inflammatory activities 195
1,8-Naphthyridines VIII. Novel 5-aminoimidazo[1,2-a][1,8]naphthyridine-6-carboxamide and 5-amino[1,2,4]triazolo[4,3-a][1,8]naphthyridine-6-carboxamide derivatives showing potent analgesic or anti-inflammatory activity, respectively, and completely devoid of acute gastrolesivity. 184
Analogs, formulations and derivatives of imatinib: A patent review 172
Synthesis, in vitro antiplatelet activity and molecular modelling studies of 10-substituted 2-(1-piperazinyl)pyrimido[1,2-a]benzimidazol-4(10H)-ones 168
1,5-Benzodiazepine tricyclic derivatives exerting anti-inflammatory effects in mice by inhibiting interleukin-6 and prostaglandin E2 production 164
1,8-Naphthyridines IV. 9-substituted N,N-dialkyl-5-(alkylamino or cycloalkylamino) [1,2,4]triazolo[4,3-a][1, 8]naphthyridine-6-carboxamides, new compounds with anti-aggressive and potent anti-inflammatory activities 163
Mechanisms involved in the antiplatelet activity of 8-methyl-4-(1-piperazinyl)-7-(3-pyridinylmethoxy)-2H-1-benzopyran-2-one (RC414) 160
Identification of new pyrrolo[2,3-d]pyrimidines as Src tyrosine kinase inhibitors in vitro active against Glioblastoma 157
1,8-Naphthyridines VI. Synthesis and anti-inflammatory activity of 5-(alkylamino)-N,N-diethyl[1,2,4]triazolo[4,3-a][1,8]naphthyridine-6 carboxamides with a new substitution pattern on the triazole ring 157
Anticonvulsive Activity in Audiogenic DBA/2 Mice of 1,4-Benzodiazepines and 1,5-Benzodiazepines with Different Activities at Cerebellar Granule Cell GABAA Receptors 157
1,5-Benzodiazepines. Part XIII. Substituted 4H-[1,2,4]triazolo[4,3-a][1,5]benzodiazepin-5-amines and 4H-imidazo[1,2-a][1,5]benzodiazepin-5-amines as analgesic, anti-inflammatory and/or antipyretic agents with low acute toxicity 155
1,5-Benzodiazepines XIV. Synthesis of new substituted 9H-bis[1,2,4]triazolo[4,3-a:3',4'-d][1,5]benzodiazepines and related compounds endowed with in vitro cytotoxic properties 152
1,8-Naphthyridines VII. New substituted 5-amino[1,2,4]triazolo[4,3-a][1,8]naphthyridine-6-carboxamides and their isosteric analogues, exhibiting notable anti-inflammatory and/or analgesic activities, but no acute gastrolesivity 151
Coumarin, chromone, and 4(3H)-pyrimidinone novel bicyclic and tricyclic derivatives as antiplatelet agents: synthesis, biological evaluation and comparative molecular field analysis 151
1,8-Naphthyridines V.Novel N-substituted 5-amino-N,N-diethyl-9-isopropyl[1,2,4]triazolo[4,3-a][1,8]naphthyridine-6-carboxamides, as potent anti-inflammatory and/or analgesic agents completely devoid of acute gastrolesivity 150
Modulation of native GABAA receptor activity by triazolo 1,5-benzodiazepines 150
New 1,5 - Benzodiazepine Compounds: Activity at Native GABAA Receptors 141
Study of the Interaction of 1,4- and 1,5-Benzodiazepines with GABAA Receptors of Rat Cerebellum Granule Cells in Culture 138
Solvent-free reactions as green chemistry procedures for the synthesis of cosmetic fatty esters 132
null 128
Conjugated Methyl Sulfide and Phenyl Sulfide Derivatives of Oxidosqualene as Inhibitors of Oxidosqualene and Squalene-Hopene Cyclases 128
Recent Studies on Ponatinib in Cancers Other Than Chronic Myeloid Leukemia 126
Pyran derivatives XX. 2-Aminochromone benzo-fused derivatives with antiproliferative properties 122
3-Cyano-4,6-diphenyl-pyridine amino acid derivatives active as influenza A polymerase inhibitors 122
Efficient one-pot synthesis of N-substituted 2-aminochromones, their benzo-fused derivatives, and diaminobenzodipyrandiones of two new structural classes 121
Synthesis of (E)- and (Z)-29-methylidyne-2,3-oxidosqualene derivatives as inhibitors of liver and yeast oxidosqualene cyclase 119
Synthesis and in vitro antiplatelet activity of new 4-(1-piperazinyl)coumarin derivatives. Human platelet phosphodiesterase 3 inhibitory properties of the two most effective compounds described and molecular modeling study on their interactions with phosphodiesterase 3A catalytic site 118
Pyrrolo[2,3-d]pyrimidines as kinase inhibitors 117
Synthesis and biological evaluation of a library of hybrid derivatives as inhibitors of influenza virus PA-PB1 interaction 117
An Update on JAK Inhibitors 117
Fine molecular tuning at position 4 of 2H-chromen-2-one derivatives in the search of potent and selective monoamine oxidase B inhibitors 114
Synthesis, antiplatelet activity and comparative molecular fields analysis of substituted 2-amino-4H-pyrido[1,2-a]pyrimidin-4-ones, their congeners and isosteric analogues 113
1,5-Benzodiazepines. Part XII. Synthesis and biological evaluation of tricyclic and tetracyclic 1,5-benzodiazepines derivatives as nevirapine analogues 111
GABA A Receptors of Cerebellar Granule in Culture: Interaction with Benzodiazepines 108
1,5-Benzodiazepines. X. Dialkylamino substituted 1,5-benzodiazepine and [1,2,4]triazolo[4,3-a][1,5]benzodiazepine derivatives with inhibitory activity on PAF-induced platelet aggregation 106
Pyran derivatives. Part XXI. Antiproliferative and cytotoxic properties of novel N-substituted 4-aminocoumarins, their benzo-fused derivatives, and some related 2-aminochromones 100
1,8-Naphthyridines III. N,N-Dialkyl-5-chloro[1,2,4]triazolo[4,3-a] [1,8]naphthyridine-6-carboxamides with anti-inflammatory activity 100
Mechanism of action of two new pyrimidoquinoline and isoquinoline derivatives in human platelets 98
Combining repositioning and de novo synthesis of pyrazolo[3,4-d]pyrimidines to discover potent SIRT-2 inhibitors 93
Acid-catalysed Hydrolisis and Benzodiazepine-like Properties of 5-(Dialkylamino)- and 5-(Alkylthio)-substituted 8-Chloro-6-phenyl-6H-[1,2,4]triazolo[4,3-a][1,5]benzodiazepines in mice 90
A family of nitrogen-containing heterocycles as sirtuin inhibitors: synthesis and invitro biological evaluation 87
Discovery of a Novel Chemo-Type for TAAR1 Agonism via Molecular Modeling 83
Anti-Survival Effect of SI306 and Its Derivatives on Human Glioblastoma Cells 82
Crystal structure of N,N-dimethyl-1-phenyl-4H-[1,2,4]triazolo[4,3-a][1,5]benzodiazepin-5-amine, C18H17N5 81
PYRAZOLO[3,4-d]PYRIMIDINE DERIVATIVES AS SIRTUIN INHIBITORS: DESIGN, SYNTHESIS AND PRELIMINARY in vitro EVALUATION 80
Sinthesis in vitro inhibitory activity on human platelet aggregation of novel properly substituted 4-(1-piperazinyl)-coumarins 75
Small Molecule Tyrosine Kinase Inhibitors (TKIs) for Glioblastoma Treatment 59
Insights into RNA-dependent RNA Polymerase Inhibitors as Anti-influenza Virus Agents 59
Synthetic Heterocyclic Derivatives as Kinase Inhibitors Tested for the Treatment of Neuroblastoma 51
Pyrazolo[3,4-d]pyrimidines as Sirtuin Inhibitors: A Preliminary Synthetic and Biological Study 44
Pyrazole[3,4-d]pyrimidine derivatives loaded into halloysite as potential CDK inhibitors 41
1,8-Naphthyridines IX. Potent anti-inflammatory and/or analgesic activity of a new group of substituted 5-amino[1,2,4]triazolo[4,3-a] [1,8]naphthyridine-6-carboxamides, of some their Mannich base derivatives and of one novel substituted 5-amino-10-oxo-10Hpyrimido[ 1,2-a][1,8]naphthyridine-6-carboxamide derivative 39
Erratum: Synthesis, antiplatelet activity and comparative molecular field analysis of substituted 2-amino-4H-pyrido[1,2-a]pyrimidin-4-ones, their congeners and isosteric analogues (Bioorganic and Medicinal Chemistry (2000) 8 (751) PII: S80968089600000109) 35
Progress of pharmaceutical technological and cosmetic research at Genoa university 23
Approaching Gallium-68 radiopharmaceuticals for tumor diagnosis: a Medicinal Chemist’s perspective 20
Halloysite Nanotube-Based Delivery of Pyrazolo[3,4-d]pyrimidine Derivatives for Prostate and Bladder Cancer Treatment 19
Synthesis, antiplatelet activity and comparative molecular field analysis of substituted 2-amino-4H-pyrido[1,2-a]pyrimidin-4-ones, their congeners and isosteric analogues 18
Evaluation of Antitumoral Activity in a 3D Cell Model of a Src Inhibitor Prodrug for Glioblastoma Treatment 12
Targeting Sirtuins with Pyrazolo[3,4-d]pyrimidines: A Synthetic and Biological Feasibility Study 12
Identification of a theranostic prodrug candidate against glioblastoma 11
Investigation the potential of SI306 SRC inhibitor and its liposomal formulation in the non-small cell lung cancer treatment 9
Investigating the potential of the SI306 Src inhibitor and its liposomal formulation in the non-small cell lung cancer treatment 9
Survivin Promotes Stem Cell Competence for Skin Cancer Initiation 2
Totale 6.649
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Categoria #
all - tutte 21.582
article - articoli 20.143
book - libri 0
conference - conferenze 1.439
curatela - curatele 0
other - altro 0
patent - brevetti 0
selected - selezionate 0
volume - volumi 0
Totale 43.164
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Totale Lug Ago Sett Ott Nov Dic Gen Feb Mar Apr Mag Giu
2020/2021262 0 0 0 22 17 50 13 33 30 46 25 26
2021/2022679 28 48 47 88 33 32 37 152 43 71 23 77
2022/2023629 56 61 6 68 79 92 3 62 89 11 90 12
2023/2024371 15 35 11 53 25 24 17 16 32 25 39 79
2024/20251.202 34 78 38 71 133 114 122 217 25 73 106 191
2025/2026742 321 62 188 171 0 0 0 0 0 0 0 0
Totale 6.649