GROSSI, GIANCARLO
GROSSI, GIANCARLO
100006 - Dipartimento di Farmacia
3-Cyano-4,6-diphenyl-pyridine amino acid derivatives active as influenza A polymerase inhibitors
2018-01-01 Giacchello, I.; Trist, I. M. L; Musumeci, F.; Greco, C.; D’Agostino, I.; Deodato, D.; Loregian, A.; Grossi, G.; Schenone, S.
A family of nitrogen-containing heterocycles as sirtuin inhibitors: synthesis and invitro biological evaluation
2024-01-01 Falesiedi, M.; Scarano, N.; Grossi, G.; Carbone, A.; Brullo, C.; Musumeci, Francesca; Bruzzone, S.; Cichero, E.; Schenone, S.
Combining repositioning and de novo synthesis of pyrazolo[3,4-d]pyrimidines to discover potent SIRT-2 inhibitors
2024-01-01 Falesiedi, Marta; Scarano, Naomi; Grossi, Giancarlo; Carbone, Anna; Brullo, Chiara; Musumeci, Francesca; Bruzzone, Santina; Cichero, Elena; Schenone, Silvia.
Identification of a theranostic prodrug candidate against glioblastoma
2025-01-01 Carbone, A.; Vagaggini, C.; Francesconi, V.; Salis, A.; Poggialini, F.; Petroni, D.; D’Antona, L.; Pozzi, C.; Grossi, G.; Tonelli, M.; Musumeci, F.; Menichetti, L.; Dreassi, E.; Schenone, S.
Investigation the potential of SI306 SRC inhibitor and its liposomal formulation in the non-small cell lung cancer treatment
2025-01-01 Poggialini, F.; Rango, E.; Vagaggini, C.; Brai, A.; Frosini, M.; Grossi, G.; Musumeci, F.; Carbone, A.; Dreassi, E.; Schenone, S.
Progress of pharmaceutical technological and cosmetic research at Genoa university
2023-01-01 Caviglioli, G.; Russo, E.; Baldassari, S.; Zuccari, G.; Ailuno, G.; Grossi, G.; Villa, C.
PYRAZOLO[3,4-d]PYRIMIDINE DERIVATIVES AS SIRTUIN INHIBITORS: DESIGN, SYNTHESIS AND PRELIMINARY in vitro EVALUATION
2024-01-01 Falesiedi, Marta; Grossi, Giancarlo; Carbone, Anna; Brullo, Chiara; Musumeci, Francesca; Bruzzone, Santina; Cichero, Elena; Schenone, Silvia
Pyrazolo[3,4-d]pyrimidines as Sirtuin Inhibitors: A Preliminary Synthetic and Biological Study
2025-01-01 Falesiedi, Marta; Scarano, Naomi; Grossi, Giancarlo; Carbone, Anna; Brullo, Chiara; Musumeci, Francesca; Bruzzone, Santina; Cichero, Elena; Schenone, Silvia
Targeting Sirtuins with Pyrazolo[3,4-d]pyrimidines: A Synthetic and Biological Feasibility Study
2025-01-01 Falesiedi, M.; Scarano, N.; Grossi, G.; Carbone, A.; Musumeci, F.; Bruzzone, Santina; Cichero, E.; Schenone, S.
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| 3-Cyano-4,6-diphenyl-pyridine amino acid derivatives active as influenza A polymerase inhibitors | 1-gen-2018 | Giacchello, I.; Trist, I. M. L; Musumeci, F.; Greco, C.; D’Agostino, I.; Deodato, D.; Loregian, A.; Grossi, G.; Schenone, S. | |
| A family of nitrogen-containing heterocycles as sirtuin inhibitors: synthesis and invitro biological evaluation | 1-gen-2024 | Falesiedi, M.; Scarano, N.; Grossi, G.; Carbone, A.; Brullo, C.; Musumeci, Francesca; Bruzzone, S.; Cichero, E.; Schenone, S. | |
| Combining repositioning and de novo synthesis of pyrazolo[3,4-d]pyrimidines to discover potent SIRT-2 inhibitors | 1-gen-2024 | Falesiedi, Marta; Scarano, Naomi; Grossi, Giancarlo; Carbone, Anna; Brullo, Chiara; Musumeci, Francesca; Bruzzone, Santina; Cichero, Elena; Schenone, Silvia. | |
| Identification of a theranostic prodrug candidate against glioblastoma | 1-gen-2025 | Carbone, A.; Vagaggini, C.; Francesconi, V.; Salis, A.; Poggialini, F.; Petroni, D.; D’Antona, L.; Pozzi, C.; Grossi, G.; Tonelli, M.; Musumeci, F.; Menichetti, L.; Dreassi, E.; Schenone, S. | |
| Investigation the potential of SI306 SRC inhibitor and its liposomal formulation in the non-small cell lung cancer treatment | 1-gen-2025 | Poggialini, F.; Rango, E.; Vagaggini, C.; Brai, A.; Frosini, M.; Grossi, G.; Musumeci, F.; Carbone, A.; Dreassi, E.; Schenone, S. | |
| Progress of pharmaceutical technological and cosmetic research at Genoa university | 1-gen-2023 | Caviglioli, G.; Russo, E.; Baldassari, S.; Zuccari, G.; Ailuno, G.; Grossi, G.; Villa, C. | |
| PYRAZOLO[3,4-d]PYRIMIDINE DERIVATIVES AS SIRTUIN INHIBITORS: DESIGN, SYNTHESIS AND PRELIMINARY in vitro EVALUATION | 1-gen-2024 | Falesiedi, Marta; Grossi, Giancarlo; Carbone, Anna; Brullo, Chiara; Musumeci, Francesca; Bruzzone, Santina; Cichero, Elena; Schenone, Silvia | |
| Pyrazolo[3,4-d]pyrimidines as Sirtuin Inhibitors: A Preliminary Synthetic and Biological Study | 1-gen-2025 | Falesiedi, Marta; Scarano, Naomi; Grossi, Giancarlo; Carbone, Anna; Brullo, Chiara; Musumeci, Francesca; Bruzzone, Santina; Cichero, Elena; Schenone, Silvia | |
| Targeting Sirtuins with Pyrazolo[3,4-d]pyrimidines: A Synthetic and Biological Feasibility Study | 1-gen-2025 | Falesiedi, M.; Scarano, N.; Grossi, G.; Carbone, A.; Musumeci, F.; Bruzzone, Santina; Cichero, E.; Schenone, S. |