IRIS
SPALLAROSSA, ANDREA
 Distribuzione geografica
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Continente #
EU - Europa 12.351
AS - Asia 48
SA - Sud America 2
NA - Nord America 1
Totale 12.402
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Nazione #
IT - Italia 12.351
CN - Cina 30
SG - Singapore 17
BR - Brasile 2
US - Stati Uniti d'America 1
VN - Vietnam 1
Totale 12.402
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Città #
Genova 6.163
Genoa 3.601
Rapallo 1.041
Vado Ligure 909
Bordighera 637
Singapore 13
Beijing 12
Ashburn 1
Blumenau 1
Ho Chi Minh City 1
Lauro de Freitas 1
Tianjin 1
Totale 12.381
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Nome #
Synthesis, SAR and molecular modelling studies of acylthiocarbamates and their parent thiocarbamates as potent non-nucleoside reverse transcriptase inhibitors related to PETT derivatives 314
Structural studies on prokaryotic sulfurtransferases 305
Studi Cristallografici di Complessi tra Transcrittasi Inversa di HIV-1 e Derivati Tiocarbammici a Scheletro Ftalimmidico, Inibitori Non Nucleosidici Correlati ai Derivati PETT. 282
A Successful Application of Parallel Synthesis to Computer-Assisted Structural Optimization of New Leads Targeting Human Immunodeficiency Virus-1 Reverse Transcriptase. The Case of Acylthiocarbamates and Thiocarbamates 169
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A persulfurated cysteine promotes active site reactivity in Azotobacter vinelandii Rhodanese 160
Further SAR studies on bicyclic basic merbarone analogues as potent antiproliferative agents 160
"One-pot" synthesis of N-acyl-N-phenylcarbamate derivatives endowed with anti-HIV and/or antiproliferative activities 155
Crystal structure of the extracellular domain of the human natural killer cell activating receptor NKp44 144
5-Substituted derivatives of 6-amino-1,3-diphenyl-2-thioxo-2,3-dihydropyrimidin-4(1H)-one as a new class of potent inhibitors of interleukin 8-induced neutrophil chemotaxis 137
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Characterization data of water-soluble hydrophilic and amphiphilic dendrimers prodrugs for delivering bioactive chemical entities otherwise non soluble. 130
Thiocarbamates as non-nucleoside HIV-1 reverse transcriptase inhibitors. Part 1: parallel synthesis, molecular modelling and structure-activity relationship studies on O-[2-(hetero)arylethyl]-N-phenylthiocarbamates 129
The three-dimensional structure of NK cell receptor NKp44, a triggering partner in natural cytotoxicity 128
Computational approaches for the design and chemical synthesis of novel F508del correctors in the treatment of cystic fibrosis 125
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X-ray analysis of HIV-1 reverse transcriptase in complex with thiocarbamates: structure-based design and synthesis of new analogues 123
Iterative design and optimization of initially inactive Proteolysis Targeting Chimeras (PROTACs) identify VZ185 as a potent, fast and selective von Hippel-Lindau (VHL)-based dual degrader probe of BRD9 and BRD7 122
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Exploring the binding features of rimonabant analogues and acyclic CB1 antagonists: docking studies and QSAR analysis 119
Unprecedented one-pot synthesis of pharmaceutical interest derivatives via in situ condensation of heterocyclic iminium salts with nitrogen nucleophiles 119
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Unprecedented one-pot stereoselective synthesis of Knoevenagel-type derivatives via in situ condensation of N-methyleniminium salts of ethylenethiourea and ethyleneurea with active methylene reagents 115
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Non-PAMAM amino acids-modified dendrimers nanoparticles for enhancing water-solubility of insoluble bioactive molecules: our state of the art 112
Anthrax toxin: structure-function relationships 111
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Thiocarbamates as non-nucleoside HIV-1 reverse transcriptase inhibitors: docking-based CoMFA and CoMSIA analyses 108
Synthesis and anti-HIV-1 activity of PETT structurally related O-substituted acyl (aryl) thiocarbamates 108
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Structure-based Design, Parallel Synthesis, SAR and Molecular Modelling Studies of Thiocarbamates, New Potent Non-Nucleoside HIV-1 Reverse Transcriptase Inhibitor Isosteres of Phenethylthiazolylthiourea Derivatives. 106
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Synthesis of indole imminun salts as key-intermediates in a convergent multi-step one-pot stereoselective synthesis of new potent antiproliferative Knoevenagel-type agent 105
Design, synthesis, SAR, and molecular modeling studies of acylthiocarbamates: a novel series of potent non-nucleoside HIV-1 reverse transcriptase inhibitors structurally related to phenethylthiazolylthiourea derivatives 105
Characterization of water soluble dendrimer formulations of an insoluble thiocarbamate derivative with moderate anti HIV-1 activity: an overview 104
Human rhinovirus 3C protease: a cysteine protease showing the trypsin(ogen)-like fold 103
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Capitolo 19 - Agenti cardiovascolari 101
The phosphoryl transfer reaction. Model of the HPr~P~IIA-Ntr protein complex 100
Insights into the Pharmacological Activity of the Imidazo-Pyrazole Scaffold 99
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Modulazioni Strutturali in O-[2-(N-Ftalimmido)etil] Acil(Aril)Tiocarbammati, Inibitori Non-Nucleosidici della Transcrittasi Inversa di HIV-1 94
Efetti della orto, meta, para sostituzione della porzione N-fenilica di O-(2-ftalimmido)etil-2-tienocarbammati sull'attività anti-HIV-1 91
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One-pot Stereoselective Synthesis of Knoevenageltype Derivatives Via Condensation of N-Methyleniminium Salts of Ethylenethiourea and Ethyleneurea with Active Methylene Reagents. 90
Capitolo 18 - Farmaci attivi sul sistema renale 90
Molecular docking of the Escherichia coli PTS system 89
Exploring the binding features of rimonabant analogues and acyclic CB1 antagonists: docking studies and 3D-QSAR analysis 89
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Studies on the catalitic activity of Azotobacter vinelandii rhodanese 88
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Modellazioni strutturali in O-[2-(N-ftalimmido)etil] Acil(Aril)tiocarbammati, inibitori non nucleosidici della trascrittasi inversa di HIV-1 86
Parallel synthesis of O-phenoxyethyl and O-adamantyl N-acyl thiocarbamates endowed with antiproliferative activity. 85
Capitolo 14 - Anticonvulsivanti 85
Sintesi parallela one-pot di disolfuri dimeri di tiocarbammati, una nuova potente classe di inibitori non nucleosidici della transcrittasi inversa 82
Btk inhibitors: a medicinal chemistry and drug delivery perspective 82
Cyclic diacyl thioureas enhance activity of corrector Lumacaftor on F508del‐CFTR 80
Non-receptor tyrosine kinase Fes as a target in oncology 78
Reattivita' di accettori di Michael atipici con nucleofili azotati 78
One-Pot Synthesis and Antiproliferative Activity of Highly Functionalized Pyrazole Derivatives 78
Regioselective Synthesis, Structural Characterization, and Antiproliferative Activity of Novel Tetra-Substituted Phenylaminopyrazole Derivatives 76
A Proteomics Approach Identifies RREB1 as a Crucial Molecular Target of Imidazo–Pyrazole Treatment in SKMEL-28 Melanoma Cells 76
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Virtual screening and structure based drug design of new Fes/Fps kinase domain inhibitors. 75
Progettazione e Sintesi di Nuovi O-[2-(N-Ftalimmido)etil]-N-(4-Cloro- e 4-Metil-Fenil)-N-Aciltiocarbammati, Inibitori Non Nucleosidici della Trancrittasi Inversa del Virus HIV-1 Attivi a Concentrazioni Nanomolari 75
Modulazioni Strutturali del Sistema Ftalimmidico di N-Aril Tiocarbammati, Inibitori Non-Nucleosidici della Transcrittasi Inversa di HIV-1 75
Synthesis and SAR studies of novel merbarone analogues 74
Synthesis and anti-HIV-1 activity of thiocarbamates, isosteres of PETT derivatives 73
Escherichia coli GlpE is a prototype sulfurtransferase for the single-domain rhodanese homology superfamily 73
Valorization and Potential Antimicrobial Use of Olive Mill Wastewater (OMW) from Italian Olive Oil Production 71
Computational studies of the binding mode and 3D-QSAR analyses of symmetric formimidoester disulfides: a new class of non-nucleoside HIV-1 reverse transcriptase inhibitors 70
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Sintesi di Esteri Tienopirimidinici ad Attività Antiproliferativa 69
Sintesi Convergente “One-Pot” di Aciltiocarbammati ad Attività Antiproliferativa 69
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Investigations of Antioxidant and Anti-Cancer Activities of 5-Aminopyrazole Derivatives 68
Mono- and di-acylated imidazolidine-2-thione derivatives: synthesis, cytotoxicity evaluation and computational studies 67
BRD9-targeting PROTACs: design, synthesis and biological evaluation 65
Potent and Broad-Spectrum Bactericidal Activity of a Nanotechnologically Manipulated Novel Pyrazole 64
Synthesis and prelimary docking studies of new colchicine-benzotriazole hybrid compounds 63
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Pharmacophore and pharmacokinetic filtering tools guiding for the design and synthesis of novel thiazole-containing and VX-809 hybrid derivatives as F508del correctors. 62
Hydrophilic and amphiphilic water-soluble dendrimer formulations of a not-soluble thiocarbamate derivative with moderate anti HIV activity for biomedical applications. 61
HIGHLY-FUNCTIONALIZED AMINO PYRAZOLES AS ANTIOXIDANT AGENTS: A PRELIMINARY SYNTHETIC ACCESSIBILITY STUDY 61
Totale 10.574
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Categoria #
all - tutte 40.746
article - articoli 24.184
book - libri 0
conference - conferenze 14.603
curatela - curatele 0
other - altro 0
patent - brevetti 0
selected - selezionate 0
volume - volumi 1.959
Totale 81.492
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Totale Lug Ago Sett Ott Nov Dic Gen Feb Mar Apr Mag Giu
2020/2021366 0 0 0 33 32 48 21 45 49 56 41 41
2021/20221.196 30 92 79 118 35 71 78 317 55 97 76 148
2022/20231.258 120 93 10 144 195 208 13 101 227 5 132 10
2023/20241.434 45 130 24 112 61 82 44 672 43 24 89 108
2024/20252.202 72 177 98 229 287 175 171 284 130 112 220 247
2025/20261.549 455 159 598 337 0 0 0 0 0 0 0 0
Totale 12.722