FOSSA, PAOLA
FOSSA, PAOLA
100006 - Dipartimento di Farmacia
2-Pyridone derivatives as inotropic agents: synthesis, pharmacology and molecular modeling study
1996-01-01 Mosti, Luisa; Boggia, Raffaella; Fossa, Paola
4-Amino-pyrazolo[3,4-d]pyrimidines with antiproliferative activity on osteosarcoma cell line SaOS-2
2005-01-01 Schenone, Silvia; Bondavalli, Francesco; Brullo, Chiara; Bruno, Olga; Ranise, A.; Mosti, L.; Menozzi, G.; Fossa, Paola; Santucci, A.; Serchi, T.; Spreafico, A.; Botta, M.
A chemometric approach to predict A1 agonist effect of adenosine analogues
2005-01-01 Fossa, Paola; Mosti, Luisa; Bondavalli, Francesco; Schenone, Silvia; Ranise, Angelo; Casolino, MARIA CHIARA; Forina, Michele
A comprehensive AIFA ligand dataset for drug repositioning
2020-01-01 Uggeri, Matteo; Rondina, Alessandro; Orro, Alessandro; D’Ursi, Pasqualina; Fossa, Paola
A water-mediated hydrogen bond network plays a crucial role in the binding affinity of PSMA radioligands
2025-01-01 Casini, Beatrice; Manconi, Andrea; Riondato, Mattia; Bauckneht, Matteo; Dighero, Edoardo; Sambuceti, Gianmario; D'Ursi, Pasqualina; Fossa, Paola
An in silico fragment-based strategy for the rational design of new glutaminase inhibitors
2025-01-01 Allahi, Shahin; Trombetti Gabriele, Antonio; Poggialini, Federica; Vagaggini, Chiara; Dreassi, Elena; Tonelli, Michele; Schenone, Silvia; Fossa, Paola; Carbone, Anna; D’Ursi, Pasqualina
Antiviral activity against ToBRFV and PepMV of Combretum micranthum leaf extracts
2022-01-01 Iobbi, V; Lanteri, Ap; Santoro, V; Minuto, G; Fossa, P; De Tommasi, N; Bisio, A
BNCT: development of a novel Boron Delivery Antibody (BDA) by means of specific residues replacement
2021-01-01 Rondina, A.; Orro, A.; Milanesi, L.; De Palma, A.; Mauri, P.; Fossa, P.; D’Ursi, P.
Characterisation of the binding pocket and drug repositioning to inhibit the interaction between the RBD spike protein of SARS-CoV-2 Omicron BA.1 and integrins
2025-01-01 Casini, Beatrice; Antonio Trombetti, Gabriele; Fossa, Paola; Zheng, Yuejuan; Bugatti, Antonella; Caruso, Arnaldo; Caccuri, Francesca; D'Ursi, Pasqualina
Computational approaches for the design and chemical synthesis of novel F508del correctors in the treatment of cystic fibrosis
2018-01-01 Righetti, Giada; Liessi, N; Pesce, E; Pedemonte, N; Salis, A; Arkel, M; Spallarossa, A; Brullo, C; Tasso, B; Damonte, G; Millo, E; Fossa, P; Cichero, E.
Computational evaluation of the synergic effect of a small molecule on Lumacaftor F508del-CFTR rescue ability
2021-01-01 Uggeri, Matteo; Orro, Alessandro; Urbinati, Chiara; Rusnati, Marco; Fossa, Paola; D’Ursi, Pasqualina
Development of a new topographical model for myocardial cGI-PDE catalytic site
1997-01-01 Fossa, Paola; Boggia, Raffaella; Mosti, Luisa
Development of new theranostic probes targeting PSMA: computational strategies to explore ligand-target interactions
2024-01-01 Casini, Beatrice; Trombetti, Gabriele; Manconi, Andrea; Riondato, Mattia; Bauckneht, Matteo; Sambuceti, Gianmario; Fossa, Paola; D’Ursi, Pasqualina
Docking and Molecular dynamics protocol for ligand binding characterization of Nuclear Receptors
2017-01-01 D’Ursi, Pasqualina; Uggeri, Matteo; Rovida, Ermanna; Fossa, Paola; Milanesi, Luciano; Orro, Alessandro
Does nicotinamide combine with lumacaftor to improve F508del-CFTR rescue?
2021-01-01 Uggeri, Matteo; Orro, Alessandro; Urbinati, Chiara; Rondina, Alessandro; Milanesi, Maria; Rusnati, Marco; D’Ursi, Pasqualina; Fossa, Paola
Efetti della orto, meta, para sostituzione della porzione N-fenilica di O-(2-ftalimmido)etil-2-tienocarbammati sull'attività anti-HIV-1
2002-01-01 Spallarossa, Andrea; Ranise, A; Bondavalli, F; Schenone, Silvia; Bruno, Olga; Fossa, Paola; Mosti, L; Menozzi, G.
Effetti della orto, meta e para Sostituzione della Porzione N-Fenilica di O-(2-Ftalimmidoetil)-2-tenoilcarbammati sull' Attività anti-HIV-1
2002-01-01 Spallarossa, Andrea; Ranise, Angelo; Bondavalli, F; Schenone, Silvia; Bruno, Olga; Fossa, Paola; Mosti, L; Menozzi, G; Marturana, F; Busonera, B; Serra, I; Cadeddu, A; Onidi, L; Poddesu, B; Loi, A. G.; LA COLLA, P.
Exploring the binding features of rimonabant analogues and acyclic CB1 antagonists: docking studies and 3D-QSAR analysis
2008-01-01 Cichero, E; Spallarossa, Andrea; Menozzi, Giulia; Mosti, Luisa; Fossa, Paola
Fragment based design of GLS1 allosteric inhibitors for cancer therapy
2025-01-01 Allahi, S.; Trombetti, G. A.; Poggialini, F.; Vagaggini, C.; Dreassi, E.; Tonelli, M.; Schenone, S.; Fossa, P.; D’Ursi, P.; Carbone, A.
Further SAR studies on bicyclic basic merbarone analogues as potent antiproliferative agents
2008-01-01 Spallarossa, Andrea; Cesarini, S; Rotolo, C; Fossa, Paola; Mosti, L; Ranise, Angelo; Sanna, G; Collu, G; Secci, B; Busonera, B; LA COLLA, P; Loddo, R.
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| 2-Pyridone derivatives as inotropic agents: synthesis, pharmacology and molecular modeling study | 1-gen-1996 | Mosti, Luisa; Boggia, Raffaella; Fossa, Paola | |
| 4-Amino-pyrazolo[3,4-d]pyrimidines with antiproliferative activity on osteosarcoma cell line SaOS-2 | 1-gen-2005 | Schenone, Silvia; Bondavalli, Francesco; Brullo, Chiara; Bruno, Olga; Ranise, A.; Mosti, L.; Menozzi, G.; Fossa, Paola; Santucci, A.; Serchi, T.; Spreafico, A.; Botta, M. | |
| A chemometric approach to predict A1 agonist effect of adenosine analogues | 1-gen-2005 | Fossa, Paola; Mosti, Luisa; Bondavalli, Francesco; Schenone, Silvia; Ranise, Angelo; Casolino, MARIA CHIARA; Forina, Michele | |
| A comprehensive AIFA ligand dataset for drug repositioning | 1-gen-2020 | Uggeri, Matteo; Rondina, Alessandro; Orro, Alessandro; D’Ursi, Pasqualina; Fossa, Paola | |
| A water-mediated hydrogen bond network plays a crucial role in the binding affinity of PSMA radioligands | 1-gen-2025 | Casini, Beatrice; Manconi, Andrea; Riondato, Mattia; Bauckneht, Matteo; Dighero, Edoardo; Sambuceti, Gianmario; D'Ursi, Pasqualina; Fossa, Paola | |
| An in silico fragment-based strategy for the rational design of new glutaminase inhibitors | 1-gen-2025 | Allahi, Shahin; Trombetti Gabriele, Antonio; Poggialini, Federica; Vagaggini, Chiara; Dreassi, Elena; Tonelli, Michele; Schenone, Silvia; Fossa, Paola; Carbone, Anna; D’Ursi, Pasqualina | |
| Antiviral activity against ToBRFV and PepMV of Combretum micranthum leaf extracts | 1-gen-2022 | Iobbi, V; Lanteri, Ap; Santoro, V; Minuto, G; Fossa, P; De Tommasi, N; Bisio, A | |
| BNCT: development of a novel Boron Delivery Antibody (BDA) by means of specific residues replacement | 1-gen-2021 | Rondina, A.; Orro, A.; Milanesi, L.; De Palma, A.; Mauri, P.; Fossa, P.; D’Ursi, P. | |
| Characterisation of the binding pocket and drug repositioning to inhibit the interaction between the RBD spike protein of SARS-CoV-2 Omicron BA.1 and integrins | 1-gen-2025 | Casini, Beatrice; Antonio Trombetti, Gabriele; Fossa, Paola; Zheng, Yuejuan; Bugatti, Antonella; Caruso, Arnaldo; Caccuri, Francesca; D'Ursi, Pasqualina | |
| Computational approaches for the design and chemical synthesis of novel F508del correctors in the treatment of cystic fibrosis | 1-gen-2018 | Righetti, Giada; Liessi, N; Pesce, E; Pedemonte, N; Salis, A; Arkel, M; Spallarossa, A; Brullo, C; Tasso, B; Damonte, G; Millo, E; Fossa, P; Cichero, E. | |
| Computational evaluation of the synergic effect of a small molecule on Lumacaftor F508del-CFTR rescue ability | 1-gen-2021 | Uggeri, Matteo; Orro, Alessandro; Urbinati, Chiara; Rusnati, Marco; Fossa, Paola; D’Ursi, Pasqualina | |
| Development of a new topographical model for myocardial cGI-PDE catalytic site | 1-gen-1997 | Fossa, Paola; Boggia, Raffaella; Mosti, Luisa | |
| Development of new theranostic probes targeting PSMA: computational strategies to explore ligand-target interactions | 1-gen-2024 | Casini, Beatrice; Trombetti, Gabriele; Manconi, Andrea; Riondato, Mattia; Bauckneht, Matteo; Sambuceti, Gianmario; Fossa, Paola; D’Ursi, Pasqualina | |
| Docking and Molecular dynamics protocol for ligand binding characterization of Nuclear Receptors | 1-gen-2017 | D’Ursi, Pasqualina; Uggeri, Matteo; Rovida, Ermanna; Fossa, Paola; Milanesi, Luciano; Orro, Alessandro | |
| Does nicotinamide combine with lumacaftor to improve F508del-CFTR rescue? | 1-gen-2021 | Uggeri, Matteo; Orro, Alessandro; Urbinati, Chiara; Rondina, Alessandro; Milanesi, Maria; Rusnati, Marco; D’Ursi, Pasqualina; Fossa, Paola | |
| Efetti della orto, meta, para sostituzione della porzione N-fenilica di O-(2-ftalimmido)etil-2-tienocarbammati sull'attività anti-HIV-1 | 1-gen-2002 | Spallarossa, Andrea; Ranise, A; Bondavalli, F; Schenone, Silvia; Bruno, Olga; Fossa, Paola; Mosti, L; Menozzi, G. | |
| Effetti della orto, meta e para Sostituzione della Porzione N-Fenilica di O-(2-Ftalimmidoetil)-2-tenoilcarbammati sull' Attività anti-HIV-1 | 1-gen-2002 | Spallarossa, Andrea; Ranise, Angelo; Bondavalli, F; Schenone, Silvia; Bruno, Olga; Fossa, Paola; Mosti, L; Menozzi, G; Marturana, F; Busonera, B; Serra, I; Cadeddu, A; Onidi, L; Poddesu, B; Loi, A. G.; LA COLLA, P. | |
| Exploring the binding features of rimonabant analogues and acyclic CB1 antagonists: docking studies and 3D-QSAR analysis | 1-gen-2008 | Cichero, E; Spallarossa, Andrea; Menozzi, Giulia; Mosti, Luisa; Fossa, Paola | |
| Fragment based design of GLS1 allosteric inhibitors for cancer therapy | 1-gen-2025 | Allahi, S.; Trombetti, G. A.; Poggialini, F.; Vagaggini, C.; Dreassi, E.; Tonelli, M.; Schenone, S.; Fossa, P.; D’Ursi, P.; Carbone, A. | |
| Further SAR studies on bicyclic basic merbarone analogues as potent antiproliferative agents | 1-gen-2008 | Spallarossa, Andrea; Cesarini, S; Rotolo, C; Fossa, Paola; Mosti, L; Ranise, Angelo; Sanna, G; Collu, G; Secci, B; Busonera, B; LA COLLA, P; Loddo, R. |