SCHENONE, SILVIA
SCHENONE, SILVIA
100006 - Dipartimento di Farmacia
(Hetero)aroyl esters of 2-(N-phthalimido)ethanol and analogues: parallel synthesis, anti-HIV-1 activity and cytotoxicity
2010-01-01 Cesarini, Sara; Spallarossa, Andrea; Ranise, Angelo; Schenone, Silvia; LA COLLA, P; Collu, G; Sanna, G; Loddo, R.
1-Acyl-, 3-acyl- and 1,3-diacyl-3-furfuryl-1-phenylthioureas with platelet antiaggregating and other activities.
1991-01-01 Ranise, Angelo; Bondavalli, Francesco; Bruno, Olga; Schenone, Silvia; Donnoli, D; Parrillo, C; Cenicola, Ml; Rossi, F.
1-Methyl and 1-(2-hydroxyalkyl)-5-(3-alkyl/cycloalkyl/phenyl/naphthylureido)-1H-pyrazole-4-carboxylic acid ethyl esters as potent human neutrophil chemotaxis inhibitors
2009-01-01 Bruno, Olga; Brullo, Chiara; Bondavalli, Francesco; Schenone, Silvia; Spisani, S; Falzarano, Ms; Varani, K; Barocelli, E; Ballabeni, V; Giorgio, C; Tognolini, M.
2-Amino/Azido/Hydrazino-5-alkoxy-5H-[1]benzopyrano[4,3-d]pyrimidines: Synthesis and Pharmacological Evaluation
2007-01-01 Bruno, Olga; Brullo, Chiara; Bondavalli, Francesco; Ranise, Angelo; Schenone, Silvia; M., Tognolini; V., Ballabeni; E., Barocelli
2-Aryl-3-phenylamino-4,5-dihydro-2h-benz[g]indazoles with analgesic activity
2003-01-01 Schenone, Silvia; Bruno, Olga; Ranise, Angelo; Brullo, Chiara; Bondavalli, Francesco; W., Filippelli; F., Mazzeo; A., Capuano; G., Falcone
2-aryl-3-phenylamino-4,5-dihydro-2H-benz[g]indazoles with antiarrhythmic and local anaesthetic activities
1995-01-01 Schenone, Silvia; Bruno, Olga; Ranise, Angelo; Bondavalli, Francesco; D'Amico, M; Filippelli, W; Falcone, G; De Novellis, V.
2-Aryl-6-methyl-3-phenylamino-6,7-dihydropyrano[4,3-c]pyrazol-4(2H)-ones with analgesic activity.
1996-01-01 Bruno, Olga; Schenone, Silvia; Ranise, Angelo; Bondavalli, Francesco; Falcone, G; Filippelli, W; Marabese, I.
2-Hydroxypropyl-β-cyclodextrin strongly improves water solubility and anti-proliferative activity of pyrazolo[3,4-d]pyrimidines Src-Abl dual inhibitors.
2010-01-01 Dreassi, E; Zizzari, At; Mori, M; Filippi, I; Belfiore, A; Naldini, A; Carraro, F; Santucci, A; Schenone, Silvia; Botta, M.
2-Phenyl-2,3-dihydro-1H-imidazo[1,2-b]pyrazole derivatives: New potent inhibitors of fMLP-induced neutrophil chemotaxis
2007-01-01 Bruno, Olga; Brullo, Chiara; Bondavalli, Francesco; Ranise, Angelo; Schenone, Silvia; Falzarano, M. S.; Varani, K; Spisani, S.
3,3-disubstituted 1-acyl-1-phenylthioureas with platelet antiaggregating and other activities
1991-01-01 Ranise, Angelo; Bondavalli, Francesco; Bruno, Olga; Schenone, Silvia; Losasso, C; Costantino, M; Cenicola, Ml; Donnoli, D; Marmo, E.
3,5-Diphenyl-1H-pyrazole derivatives. XII. N-substituted 4-amino-1-(2-hydroxy- or 2-alkylaminoethyl)-3,5-diphenyl-1H-pyrazoles with local anesthetic, analgesic and platelet antiaggregating activities.
1994-01-01 Bruno, Olga; Ranise, Angelo; Bondavalli, Francesco; Schenone, Silvia; D'Amico, M; Falciani, M; Vacca, C; Filippelli, A.
3-(Arylamino)-6,7-dihydro-6-methylpyrano[4,3-c]pyrazol-4(1H or 2H)-ones with antipyretic, analgesic, antiarrhythmic, hypotensive and other activities.
1993-01-01 Bruno, Olga; Ranise, Angelo; Schenone, Silvia; Bondavalli, Francesco; D'Amico, M; Falciani, M; Berrino, L; Rossi, F.
3-Arylsulphonyl-5-arylamino-1,3,4-thiadiazol-2(3H)ones as antiinflammatory and analgesic agents
2001-01-01 Schenone, Silvia; Bruno, Olga; Ranise, Angelo; Bondavalli, Francesco; Filippelli, W; Falcone, G; Giordano, L; Vitelli, M. R.
3D QSAR models built on structure-based alignments of Abl tyrosine kinase inhibitors.
2009-01-01 F., Falchi; F., Manetti; F., Carraro; A., Naldini; G., Maga; E., Crespan; Schenone, Silvia; Bruno, Olga; Brullo, Chiara; M. Botta, .
4-Amino-Substituted Pyrazolo[3,4-d]Pyrimidines: Synthesis and Biological Properties
2009-01-01 Schenone, S.; Bruno, O.; Radi, M.; Botta, M.
5-[[ω-(Dialkylamino)alkoxy]methylene]-1,3,3-trimethyl-2-oxabicyclo[2.2.2]octan-6-ones with hypotensive, local anesthetic, antiarrhythmic and other activities
1994-01-01 Schenone, Silvia; Bruno, Olga; Ranise, Angelo; Bondavalli, Francesco; D'Amico, M; Piu, M; Filippelli, W; Berrino, L.
5-Substituted 2,3-dihydro-6-mercapto-1,3-diphenyl-2-thioxo-4(3H)-pyrimidinones and their 6-(acylthio) derivatives with platelet antiaggregating, antiinflammatory, antiarrhythmic, antihyperlipidemic and other activities.
1994-01-01 Ranise, Angelo; Bruno, Olga; Bondavalli, Francesco; Schenone, Silvia; D'Amico, M; Falciani, M; Filippelli, W; Rossi, F.
A cascade screening approach for the identification of Bcr-Abl myristate pocket binders active against wild type and T315I mutant
2016-01-01 Radi, Marco; Schneider, Ralf; Fallacara, Anna Lucia; Botta, Lorenzo; Crespan, Emmanuele; Tintori, Cristina; Maga, Giovanni; Kissova, Miroslava; Calgani, Alessia; Richters, André; Musumeci, Francesca; Rauh, Daniel; Schenone, Silvia
A class of pyrrole derivatives endowed with analgesic/anti-inflammatory activity.
2013-01-01 Battilocchio, C; Poce, G; Alfonso, S; Porretta, Gc; Consalvi, S; Sautebin, L; Pace, S; Rossi, A; Ghelardini, C; Di Cesare Mannelli, L; Schenone, Silvia; Giordani, A; Di Francesco, L; Patrignani, P; Biava, M.
A combination of docking/dynamics simulations and pharmacophoric modeling to discover new dual c-Src/Abl kinase inhibitors.
2006-01-01 Manetti, F; Locatelli, Ga; Maga, G; Schenone, Silvia; Modugno, M; Forli, S; Corelli, F; Botta, M.
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| (Hetero)aroyl esters of 2-(N-phthalimido)ethanol and analogues: parallel synthesis, anti-HIV-1 activity and cytotoxicity | 1-gen-2010 | Cesarini, Sara; Spallarossa, Andrea; Ranise, Angelo; Schenone, Silvia; LA COLLA, P; Collu, G; Sanna, G; Loddo, R. | |
| 1-Acyl-, 3-acyl- and 1,3-diacyl-3-furfuryl-1-phenylthioureas with platelet antiaggregating and other activities. | 1-gen-1991 | Ranise, Angelo; Bondavalli, Francesco; Bruno, Olga; Schenone, Silvia; Donnoli, D; Parrillo, C; Cenicola, Ml; Rossi, F. | |
| 1-Methyl and 1-(2-hydroxyalkyl)-5-(3-alkyl/cycloalkyl/phenyl/naphthylureido)-1H-pyrazole-4-carboxylic acid ethyl esters as potent human neutrophil chemotaxis inhibitors | 1-gen-2009 | Bruno, Olga; Brullo, Chiara; Bondavalli, Francesco; Schenone, Silvia; Spisani, S; Falzarano, Ms; Varani, K; Barocelli, E; Ballabeni, V; Giorgio, C; Tognolini, M. | |
| 2-Amino/Azido/Hydrazino-5-alkoxy-5H-[1]benzopyrano[4,3-d]pyrimidines: Synthesis and Pharmacological Evaluation | 1-gen-2007 | Bruno, Olga; Brullo, Chiara; Bondavalli, Francesco; Ranise, Angelo; Schenone, Silvia; M., Tognolini; V., Ballabeni; E., Barocelli | |
| 2-Aryl-3-phenylamino-4,5-dihydro-2h-benz[g]indazoles with analgesic activity | 1-gen-2003 | Schenone, Silvia; Bruno, Olga; Ranise, Angelo; Brullo, Chiara; Bondavalli, Francesco; W., Filippelli; F., Mazzeo; A., Capuano; G., Falcone | |
| 2-aryl-3-phenylamino-4,5-dihydro-2H-benz[g]indazoles with antiarrhythmic and local anaesthetic activities | 1-gen-1995 | Schenone, Silvia; Bruno, Olga; Ranise, Angelo; Bondavalli, Francesco; D'Amico, M; Filippelli, W; Falcone, G; De Novellis, V. | |
| 2-Aryl-6-methyl-3-phenylamino-6,7-dihydropyrano[4,3-c]pyrazol-4(2H)-ones with analgesic activity. | 1-gen-1996 | Bruno, Olga; Schenone, Silvia; Ranise, Angelo; Bondavalli, Francesco; Falcone, G; Filippelli, W; Marabese, I. | |
| 2-Hydroxypropyl-β-cyclodextrin strongly improves water solubility and anti-proliferative activity of pyrazolo[3,4-d]pyrimidines Src-Abl dual inhibitors. | 1-gen-2010 | Dreassi, E; Zizzari, At; Mori, M; Filippi, I; Belfiore, A; Naldini, A; Carraro, F; Santucci, A; Schenone, Silvia; Botta, M. | |
| 2-Phenyl-2,3-dihydro-1H-imidazo[1,2-b]pyrazole derivatives: New potent inhibitors of fMLP-induced neutrophil chemotaxis | 1-gen-2007 | Bruno, Olga; Brullo, Chiara; Bondavalli, Francesco; Ranise, Angelo; Schenone, Silvia; Falzarano, M. S.; Varani, K; Spisani, S. | |
| 3,3-disubstituted 1-acyl-1-phenylthioureas with platelet antiaggregating and other activities | 1-gen-1991 | Ranise, Angelo; Bondavalli, Francesco; Bruno, Olga; Schenone, Silvia; Losasso, C; Costantino, M; Cenicola, Ml; Donnoli, D; Marmo, E. | |
| 3,5-Diphenyl-1H-pyrazole derivatives. XII. N-substituted 4-amino-1-(2-hydroxy- or 2-alkylaminoethyl)-3,5-diphenyl-1H-pyrazoles with local anesthetic, analgesic and platelet antiaggregating activities. | 1-gen-1994 | Bruno, Olga; Ranise, Angelo; Bondavalli, Francesco; Schenone, Silvia; D'Amico, M; Falciani, M; Vacca, C; Filippelli, A. | |
| 3-(Arylamino)-6,7-dihydro-6-methylpyrano[4,3-c]pyrazol-4(1H or 2H)-ones with antipyretic, analgesic, antiarrhythmic, hypotensive and other activities. | 1-gen-1993 | Bruno, Olga; Ranise, Angelo; Schenone, Silvia; Bondavalli, Francesco; D'Amico, M; Falciani, M; Berrino, L; Rossi, F. | |
| 3-Arylsulphonyl-5-arylamino-1,3,4-thiadiazol-2(3H)ones as antiinflammatory and analgesic agents | 1-gen-2001 | Schenone, Silvia; Bruno, Olga; Ranise, Angelo; Bondavalli, Francesco; Filippelli, W; Falcone, G; Giordano, L; Vitelli, M. R. | |
| 3D QSAR models built on structure-based alignments of Abl tyrosine kinase inhibitors. | 1-gen-2009 | F., Falchi; F., Manetti; F., Carraro; A., Naldini; G., Maga; E., Crespan; Schenone, Silvia; Bruno, Olga; Brullo, Chiara; M. Botta, . | |
| 4-Amino-Substituted Pyrazolo[3,4-d]Pyrimidines: Synthesis and Biological Properties | 1-gen-2009 | Schenone, S.; Bruno, O.; Radi, M.; Botta, M. | |
| 5-[[ω-(Dialkylamino)alkoxy]methylene]-1,3,3-trimethyl-2-oxabicyclo[2.2.2]octan-6-ones with hypotensive, local anesthetic, antiarrhythmic and other activities | 1-gen-1994 | Schenone, Silvia; Bruno, Olga; Ranise, Angelo; Bondavalli, Francesco; D'Amico, M; Piu, M; Filippelli, W; Berrino, L. | |
| 5-Substituted 2,3-dihydro-6-mercapto-1,3-diphenyl-2-thioxo-4(3H)-pyrimidinones and their 6-(acylthio) derivatives with platelet antiaggregating, antiinflammatory, antiarrhythmic, antihyperlipidemic and other activities. | 1-gen-1994 | Ranise, Angelo; Bruno, Olga; Bondavalli, Francesco; Schenone, Silvia; D'Amico, M; Falciani, M; Filippelli, W; Rossi, F. | |
| A cascade screening approach for the identification of Bcr-Abl myristate pocket binders active against wild type and T315I mutant | 1-gen-2016 | Radi, Marco; Schneider, Ralf; Fallacara, Anna Lucia; Botta, Lorenzo; Crespan, Emmanuele; Tintori, Cristina; Maga, Giovanni; Kissova, Miroslava; Calgani, Alessia; Richters, André; Musumeci, Francesca; Rauh, Daniel; Schenone, Silvia | |
| A class of pyrrole derivatives endowed with analgesic/anti-inflammatory activity. | 1-gen-2013 | Battilocchio, C; Poce, G; Alfonso, S; Porretta, Gc; Consalvi, S; Sautebin, L; Pace, S; Rossi, A; Ghelardini, C; Di Cesare Mannelli, L; Schenone, Silvia; Giordani, A; Di Francesco, L; Patrignani, P; Biava, M. | |
| A combination of docking/dynamics simulations and pharmacophoric modeling to discover new dual c-Src/Abl kinase inhibitors. | 1-gen-2006 | Manetti, F; Locatelli, Ga; Maga, G; Schenone, Silvia; Modugno, M; Forli, S; Corelli, F; Botta, M. |