LUSARDI, MATTEO
LUSARDI, MATTEO
100006 - Dipartimento di Farmacia
Amino-Pyrazoles in Medicinal Chemistry: A Review
2023-01-01 Lusardi, Matteo; Spallarossa, Andrea; Brullo, Chiara
Antimalarial Activity of Tri- and Tetra-Substituted Anilino Pyrazoles
2023-01-01 Lusardi, Matteo; Basilico, Nicoletta; Rotolo, Chiara; Parapini, Silvia; Spallarossa, Andrea
Antiprotozoal Activity of Highly Substituted Pyrazole and Pyrimidine Derivatives
2025-01-01 Lusardi, M.; Basilico, N.; Iervasi, E.; Brullo, C.; Parapini, S.; Ponassi, M.; Rosano, C.; Spallarossa, A.
Bicyclic basic merbarone analogues as antiproliferative agents
2021-01-01 Spallarossa, A.; Lusardi, M.; Caneva, C.; Profumo, A.; Rosano, C.; Ponassi, M.
Cyclic diacyl thioureas enhance activity of corrector Lumacaftor on F508del‐CFTR
2024-01-01 Spallarossa, Andrea; Pedemonte, Nicoletta; Pesce, Emanuela; Millo, Enrico; Cichero, Elena; Rosano, Camillo; Lusardi, Matteo; Iervasi, Erika; Ponassi, Marco
Novel 5-aminopyrazoles endowed with anti-angiogenetic properties: Design, synthesis and biological evaluation
2023-01-01 Lusardi, Matteo; Wehrle-Haller, Bernhard; Sidibe, Adama; Ponassi, Marco; Iervasi, Erika; Rosano, Camillo; Brullo, Chiara; Spallarossa, Andrea
Novel tetrasubstituted 5-Arylamino pyrazoles able to interfere with angiogenesis and Ca2+ mobilization
2024-01-01 Lusardi, Matteo; Belvedere, Raffaella; Petrella, Antonello; Iervasi, Erika; Ponassi, Marco; Brullo, Chiara; Spallarossa, Andrea
One-Pot Synthesis and Antiproliferative Activity of Highly Functionalized Pyrazole Derivatives
2022-01-01 Lusardi, M.; Rotolo, C.; Ponassi, M.; Iervasi, E.; Rosano, C.; Spallarossa, A.
PDE4D: A Multipurpose Pharmacological Target
2024-01-01 Lusardi, Matteo; Rapetti, Federica; Spallarossa, Andrea; Brullo, Chiara
Potent and Broad-Spectrum Bactericidal Activity of a Nanotechnologically Manipulated Novel Pyrazole
2022-01-01 Alfei, Silvana; Caviglia, Debora; Zorzoli, Alessia; Marimpietri, Danilo; Spallarossa, Andrea; Lusardi, Matteo; Zuccari, Guendalina; Schito, Anna Maria
Regioselective Synthesis, Structural Characterization, and Antiproliferative Activity of Novel Tetra-Substituted Phenylaminopyrazole Derivatives
2022-01-01 Lusardi, Matteo; Profumo, Aldo; Rotolo, Chiara; Iervasi, Erika; Rosano, Camillo; Spallarossa, Andrea; Ponassi, Marco
Scouting in silico different chemo-types of PDE4 inhibitors to guide the design of new anti-inflammatory/antioxidant agents
2023-01-01 Cichero, Elena; Rapetti, Federica; Lusardi, Matteo; Scarano, Naomi; Alfei, Silvana; Altieri, Paola; Garibaldi, Silvano; Ameri, Pietro; Signorello, MARIA GRAZIA; Brullo, Chiara
Structure–Activity Relationship Studies on Highly Functionalized Pyrazole Hydrazones and Amides as Antiproliferative and Antioxidant Agents
2024-01-01 Lusardi, Matteo; Signorello, Maria Grazia; Russo, Eleonora; Caviglia, Debora; Ponassi, Marco; Iervasi, Erika; Rosano, Camillo; Brullo, Chiara; Spallarossa, Andrea
Successful Dendrimer and Liposome-Based Strategies to Solubilize an Antiproliferative Pyrazole Otherwise Not Clinically Applicable
2022-01-01 Alfei, S.; Spallarossa, A.; Lusardi, M.; Zuccari, G.
Targeting Ubiquitin‐Specific Protease 7 with Novel 5‐Amino‐Pyrazole Inhibitors: Design, Synthesis, and Biological Evaluation
2025-01-01 Lusardi, Matteo; Morretta, Elva; Spallarossa, Andrea; Chiara Monti, Maria; Rosano, Camillo; Iervasi, Erika; Ponassi, Marco; Mori, Matteo; Meneghetti, Fiorella; Brullo, Chiara
Triazole-imidazo[1,2-b]pyrazoles Able to Counteract Melanoma Cell Survival Without Compromising the Viability of Healthy Keratinocytes
2025-01-01 Brullo, Chiara; Marengo, Barbara; Domenicotti, Cinzia; Lusardi, Matteo; Cichero, Elena; Salis, Annalisa; Caviglia, Debora; Russo, Eleonora; Spallarossa, Andrea
USP7 at the Crossroads of Ubiquitin Signaling, Cell Cycle, and Tumorigenesis
2025-01-01 Lusardi, Matteo; Rapetti, Federica; Spallarossa, Andrea; Massone, Marta; Cichero, Elena; Brullo, Chiara
| Titolo | Data di pubblicazione | Autore(i) | File |
|---|---|---|---|
| Amino-Pyrazoles in Medicinal Chemistry: A Review | 1-gen-2023 | Lusardi, Matteo; Spallarossa, Andrea; Brullo, Chiara | |
| Antimalarial Activity of Tri- and Tetra-Substituted Anilino Pyrazoles | 1-gen-2023 | Lusardi, Matteo; Basilico, Nicoletta; Rotolo, Chiara; Parapini, Silvia; Spallarossa, Andrea | |
| Antiprotozoal Activity of Highly Substituted Pyrazole and Pyrimidine Derivatives | 1-gen-2025 | Lusardi, M.; Basilico, N.; Iervasi, E.; Brullo, C.; Parapini, S.; Ponassi, M.; Rosano, C.; Spallarossa, A. | |
| Bicyclic basic merbarone analogues as antiproliferative agents | 1-gen-2021 | Spallarossa, A.; Lusardi, M.; Caneva, C.; Profumo, A.; Rosano, C.; Ponassi, M. | |
| Cyclic diacyl thioureas enhance activity of corrector Lumacaftor on F508del‐CFTR | 1-gen-2024 | Spallarossa, Andrea; Pedemonte, Nicoletta; Pesce, Emanuela; Millo, Enrico; Cichero, Elena; Rosano, Camillo; Lusardi, Matteo; Iervasi, Erika; Ponassi, Marco | |
| Novel 5-aminopyrazoles endowed with anti-angiogenetic properties: Design, synthesis and biological evaluation | 1-gen-2023 | Lusardi, Matteo; Wehrle-Haller, Bernhard; Sidibe, Adama; Ponassi, Marco; Iervasi, Erika; Rosano, Camillo; Brullo, Chiara; Spallarossa, Andrea | |
| Novel tetrasubstituted 5-Arylamino pyrazoles able to interfere with angiogenesis and Ca2+ mobilization | 1-gen-2024 | Lusardi, Matteo; Belvedere, Raffaella; Petrella, Antonello; Iervasi, Erika; Ponassi, Marco; Brullo, Chiara; Spallarossa, Andrea | |
| One-Pot Synthesis and Antiproliferative Activity of Highly Functionalized Pyrazole Derivatives | 1-gen-2022 | Lusardi, M.; Rotolo, C.; Ponassi, M.; Iervasi, E.; Rosano, C.; Spallarossa, A. | |
| PDE4D: A Multipurpose Pharmacological Target | 1-gen-2024 | Lusardi, Matteo; Rapetti, Federica; Spallarossa, Andrea; Brullo, Chiara | |
| Potent and Broad-Spectrum Bactericidal Activity of a Nanotechnologically Manipulated Novel Pyrazole | 1-gen-2022 | Alfei, Silvana; Caviglia, Debora; Zorzoli, Alessia; Marimpietri, Danilo; Spallarossa, Andrea; Lusardi, Matteo; Zuccari, Guendalina; Schito, Anna Maria | |
| Regioselective Synthesis, Structural Characterization, and Antiproliferative Activity of Novel Tetra-Substituted Phenylaminopyrazole Derivatives | 1-gen-2022 | Lusardi, Matteo; Profumo, Aldo; Rotolo, Chiara; Iervasi, Erika; Rosano, Camillo; Spallarossa, Andrea; Ponassi, Marco | |
| Scouting in silico different chemo-types of PDE4 inhibitors to guide the design of new anti-inflammatory/antioxidant agents | 1-gen-2023 | Cichero, Elena; Rapetti, Federica; Lusardi, Matteo; Scarano, Naomi; Alfei, Silvana; Altieri, Paola; Garibaldi, Silvano; Ameri, Pietro; Signorello, MARIA GRAZIA; Brullo, Chiara | |
| Structure–Activity Relationship Studies on Highly Functionalized Pyrazole Hydrazones and Amides as Antiproliferative and Antioxidant Agents | 1-gen-2024 | Lusardi, Matteo; Signorello, Maria Grazia; Russo, Eleonora; Caviglia, Debora; Ponassi, Marco; Iervasi, Erika; Rosano, Camillo; Brullo, Chiara; Spallarossa, Andrea | |
| Successful Dendrimer and Liposome-Based Strategies to Solubilize an Antiproliferative Pyrazole Otherwise Not Clinically Applicable | 1-gen-2022 | Alfei, S.; Spallarossa, A.; Lusardi, M.; Zuccari, G. | |
| Targeting Ubiquitin‐Specific Protease 7 with Novel 5‐Amino‐Pyrazole Inhibitors: Design, Synthesis, and Biological Evaluation | 1-gen-2025 | Lusardi, Matteo; Morretta, Elva; Spallarossa, Andrea; Chiara Monti, Maria; Rosano, Camillo; Iervasi, Erika; Ponassi, Marco; Mori, Matteo; Meneghetti, Fiorella; Brullo, Chiara | |
| Triazole-imidazo[1,2-b]pyrazoles Able to Counteract Melanoma Cell Survival Without Compromising the Viability of Healthy Keratinocytes | 1-gen-2025 | Brullo, Chiara; Marengo, Barbara; Domenicotti, Cinzia; Lusardi, Matteo; Cichero, Elena; Salis, Annalisa; Caviglia, Debora; Russo, Eleonora; Spallarossa, Andrea | |
| USP7 at the Crossroads of Ubiquitin Signaling, Cell Cycle, and Tumorigenesis | 1-gen-2025 | Lusardi, Matteo; Rapetti, Federica; Spallarossa, Andrea; Massone, Marta; Cichero, Elena; Brullo, Chiara |